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Compound
PGDB_C002827
8 activity records1 related patents
2D structure
COc1ccc(Oc2ccc(C(=O)Nc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)cc2)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 6.5 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A013617 | PGDB_C002827 | PGDB_AS000707 | View |
| % Degradation | - | = | 84.5 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A024589 | PGDB_C002827 | PGDB_AS000892 | View |
| % Degradation | - | = | 16.2 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A037091 | PGDB_C002827 | PGDB_AS000768 | View |
| % Degradation | - | = | 53.6 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A046632 | PGDB_C002827 | PGDB_AS001414 | View |
| % Degradation | - | = | 4.8 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A052100 | PGDB_C002827 | PGDB_AS001974 | View |
| % Degradation | - | = | 55.8 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A060620 | PGDB_C002827 | PGDB_AS000685 | View |
| % Degradation | - | = | 44.9 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A073147 | PGDB_C002827 | PGDB_AS000209 | View |
| % Degradation | - | = | 4.3 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A075192 | PGDB_C002827 | PGDB_AS002431 | View |