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Compound
PGDB_C002839
8 activity records1 related patents
2D structure
COc1cc(Br)cc2c1OCC(C(=O)Nc1ccc3c(c1)CN(C1CCC(=O)NC1=O)C3=O)=C2Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 1.6 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A015556 | PGDB_C002839 | PGDB_AS002431 | View |
| % Degradation | - | = | 87.8 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A035309 | PGDB_C002839 | PGDB_AS000892 | View |
| % Degradation | - | = | 64.7 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A043744 | PGDB_C002839 | PGDB_AS000209 | View |
| % Degradation | - | = | 12.6 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A045616 | PGDB_C002839 | PGDB_AS000707 | View |
| % Degradation | - | = | 4.1 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A060134 | PGDB_C002839 | PGDB_AS001974 | View |
| % Degradation | - | = | 74.4 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A067838 | PGDB_C002839 | PGDB_AS001414 | View |
| % Degradation | - | = | 26.1 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A070253 | PGDB_C002839 | PGDB_AS000768 | View |
| % Degradation | - | = | 68 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A076230 | PGDB_C002839 | PGDB_AS000685 | View |