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Compound
PGDB_C002840
8 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(NC(=O)C4=Cc5cc(Br)cc(Br)c5OC4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 46.5 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A023142 | PGDB_C002840 | PGDB_AS000209 | View |
| % Degradation | - | = | 12.3 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A032074 | PGDB_C002840 | PGDB_AS000707 | View |
| % Degradation | - | = | 62.6 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A036181 | PGDB_C002840 | PGDB_AS000892 | View |
| % Degradation | - | = | 5.3 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A044645 | PGDB_C002840 | PGDB_AS002431 | View |
| % Degradation | - | = | 48.7 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A054551 | PGDB_C002840 | PGDB_AS001414 | View |
| % Degradation | - | = | 54.7 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A057140 | PGDB_C002840 | PGDB_AS000685 | View |
| % Degradation | - | = | 9.2 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A057413 | PGDB_C002840 | PGDB_AS001974 | View |
| % Degradation | - | = | 22.6 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A069391 | PGDB_C002840 | PGDB_AS000768 | View |