Assay

PGDB_AS002492

System: cell_basedTarget: GSPT1Cell line: HEK293
Assay context summary

Assay context

22 activity records
Assay family% Degradation
Systemcell_based
ReadoutEC50
TargetGSPT1
E3Not specified
Cell lineHEK293
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

22 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C008163
EC50-=253nM-—GSPT1-HEK293IL323841APGDB_A007222PGDB_C008163PGDB_AS002492View
2D structure for PGDB_C008166
EC50-=68.4nM-—GSPT1-HEK293IL323841APGDB_A008332PGDB_C008166PGDB_AS002492View
2D structure for PGDB_C008164
EC50-=153nM-—GSPT1-HEK293IL323841APGDB_A011074PGDB_C008164PGDB_AS002492View
2D structure for PGDB_C001361
EC50-=198.3nM-—GSPT1-HEK293IL323841APGDB_A012632PGDB_C001361PGDB_AS002492View
2D structure for PGDB_C008162
EC50-=144.9nM-—GSPT1-HEK293IL323841APGDB_A013905PGDB_C008162PGDB_AS002492View
2D structure for PGDB_C008154
EC50-=87.1nM-—GSPT1-HEK293IL323841APGDB_A015734PGDB_C008154PGDB_AS002492View
2D structure for PGDB_C008159
EC50-=337nM-—GSPT1-HEK293IL323841APGDB_A019451PGDB_C008159PGDB_AS002492View
2D structure for PGDB_C008155
EC50-=288nM-—GSPT1-HEK293IL323841APGDB_A020369PGDB_C008155PGDB_AS002492View
2D structure for PGDB_C008152
EC50-=128.4nM-—GSPT1-HEK293IL323841APGDB_A026071PGDB_C008152PGDB_AS002492View
2D structure for PGDB_C008161
EC50-=289nM-—GSPT1-HEK293IL323841APGDB_A026745PGDB_C008161PGDB_AS002492View
2D structure for PGDB_C008168
EC50-=94.1nM-—GSPT1-HEK293IL323841APGDB_A031642PGDB_C008168PGDB_AS002492View
2D structure for PGDB_C019545
EC50-=506nM-—GSPT1-HEK293IL323841APGDB_A032802PGDB_C019545PGDB_AS002492View
2D structure for PGDB_C008167
EC50-=123nM-—GSPT1-HEK293IL323841APGDB_A040779PGDB_C008167PGDB_AS002492View
2D structure for PGDB_C008160
EC50-=2590nM-—GSPT1-HEK293IL323841APGDB_A046605PGDB_C008160PGDB_AS002492View
2D structure for PGDB_C008158
EC50-=2080nM-—GSPT1-HEK293IL323841APGDB_A053018PGDB_C008158PGDB_AS002492View
2D structure for PGDB_C008150
EC50-=140nM-—GSPT1-HEK293IL323841APGDB_A053889PGDB_C008150PGDB_AS002492View
2D structure for PGDB_C008156
EC50-=731nM-—GSPT1-HEK293IL323841APGDB_A062693PGDB_C008156PGDB_AS002492View
2D structure for PGDB_C008157
EC50-=99.2nM-—GSPT1-HEK293IL323841APGDB_A063932PGDB_C008157PGDB_AS002492View
2D structure for PGDB_C008153
EC50-=116nM-—GSPT1-HEK293IL323841APGDB_A064902PGDB_C008153PGDB_AS002492View
2D structure for PGDB_C008149
EC50-=216.8nM-—GSPT1-HEK293IL323841APGDB_A066520PGDB_C008149PGDB_AS002492View
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