Summary
AssigneeBeijing Innocare Pharma Tech
Filing years2024
Patents2
Compounds77
Activity records208
Patent families2
Targets1
Assay familiesdegradation, viability
Activity metricsDC50, Dmax, GI50, IC50
Overview

Target distribution and active-compound trend

Target distribution

208 activity records

1 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

0224420242025
Activity compounds and values

Activity records

208 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C003182
DC50-=7.2nM-GSPT1-NB4WO2024222614A1PGDB_A007290PGDB_C003182PGDB_AS001663View
2D structure for PGDB_C003214
GI50-=22nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A007848PGDB_C003214PGDB_AS000187View
2D structure for PGDB_C003200
DC50->1000nM-GSPT1-NB4WO2024222614A1PGDB_A008465PGDB_C003200PGDB_AS001663View
2D structure for PGDB_C003217
Dmax-=125%--GSPT1-NB4WO2024222614A1PGDB_A008622PGDB_C003217PGDB_AS000251View
2D structure for PGDB_C003210
GI50-=39nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A009532PGDB_C003210PGDB_AS000187View
2D structure for PGDB_C003186
Dmax-=112%--GSPT1-NB4WO2024222614A1PGDB_A010052PGDB_C003186PGDB_AS000251View
2D structure for PGDB_C003197
DC50-=15nM-GSPT1-NB4WO2024222614A1PGDB_A013016PGDB_C003197PGDB_AS001663View
2D structure for PGDB_C003183
GI50-=35nM-GSPT1-NB4WO2024222614A1PGDB_A013366PGDB_C003183PGDB_AS001086View
2D structure for PGDB_C003181
Dmax-=94%--GSPT1-NB4WO2024222614A1PGDB_A013551PGDB_C003181PGDB_AS000251View
2D structure for PGDB_C003184
GI50-=4.5nM-GSPT1-NB4WO2024222614A1PGDB_A014707PGDB_C003184PGDB_AS001086View
2D structure for PGDB_C003184
Dmax-=113%--GSPT1-NB4WO2024222614A1PGDB_A015376PGDB_C003184PGDB_AS000251View
2D structure for PGDB_C003175
GI50-=33nM-GSPT1-NB4WO2024222614A1PGDB_A016267PGDB_C003175PGDB_AS001086View
2D structure for PGDB_C003207
GI50-=10nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A017336PGDB_C003207PGDB_AS000187View
2D structure for PGDB_C003196
Dmax-=16%--GSPT1-NB4WO2024222614A1PGDB_A017501PGDB_C003196PGDB_AS000251View
2D structure for PGDB_C003201
DC50-=4.8nM-GSPT1-NB4WO2024222614A1PGDB_A019557PGDB_C003201PGDB_AS001663View
2D structure for PGDB_C003181
GI50-=23nM-GSPT1-NB4WO2024222614A1PGDB_A019808PGDB_C003181PGDB_AS001086View
2D structure for PGDB_C003190
GI50-=23nM-GSPT1-NB4WO2024222614A1PGDB_A022412PGDB_C003190PGDB_AS001086View
2D structure for PGDB_C003181
DC50-=5.2nM-GSPT1-NB4WO2024222614A1PGDB_A023306PGDB_C003181PGDB_AS001663View
2D structure for PGDB_C003177
DC50->1000nM-GSPT1-NB4WO2024222614A1PGDB_A023514PGDB_C003177PGDB_AS001663View
2D structure for PGDB_C003216
GI50-=19nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A023941PGDB_C003216PGDB_AS000187View