Summary
AssigneeZhuhai Woo Biological Science And Technology
Filing years2023
Patents1
Compounds114
Activity records229
Patent families1
Targets1
Assay familiesdegradation, viability
Activity metricsDC50, GI50
Overview

Target distribution and active-compound trend

Target distribution

229 activity records

1 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

0571142025
Activity compounds and values

Activity records

229 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C002250
GI50-<100nM-GSPT1-HL-60WO2023237116A1PGDB_A008007PGDB_C002250PGDB_AS001555View
2D structure for PGDB_C002259
GI50-=22.29nM-GSPT1-Hep3BWO2023237116A1PGDB_A009004PGDB_C002259PGDB_AS001914View
2D structure for PGDB_C002253
DC50-<100nM-GSPT1-HEK293WO2023237116A1PGDB_A009125PGDB_C002253PGDB_AS002200View
2D structure for PGDB_C002274
DC50-<100nM-GSPT1-HEK293WO2023237116A1PGDB_A009352PGDB_C002274PGDB_AS002200View
2D structure for PGDB_C002266
DC50-<100nM-GSPT1-HEK293WO2023237116A1PGDB_A009563PGDB_C002266PGDB_AS002200View
2D structure for PGDB_C002214
DC50-<100nM-GSPT1-HEK293WO2023237116A1PGDB_A010038PGDB_C002214PGDB_AS002200View
2D structure for PGDB_C002237
DC50-<100nM-GSPT1-HEK293WO2023237116A1PGDB_A010570PGDB_C002237PGDB_AS002200View
2D structure for PGDB_C002206
DC50-<100nM-GSPT1-HEK293WO2023237116A1PGDB_A010862PGDB_C002206PGDB_AS002200View
2D structure for PGDB_C002248
GI50-=100-1000nM-GSPT1-HL-60WO2023237116A1PGDB_A011190PGDB_C002248PGDB_AS001555View
2D structure for PGDB_C002298
GI50-<100nM-GSPT1-HL-60WO2023237116A1PGDB_A011499PGDB_C002298PGDB_AS001555View
2D structure for PGDB_C002260
DC50-<100nM-GSPT1-HEK293WO2023237116A1PGDB_A011994PGDB_C002260PGDB_AS002200View
2D structure for PGDB_C002256
GI50-<100nM-GSPT1-HL-60WO2023237116A1PGDB_A012098PGDB_C002256PGDB_AS001555View
2D structure for PGDB_C002245
DC50-=100-1000nM-GSPT1-HEK293WO2023237116A1PGDB_A012610PGDB_C002245PGDB_AS002200View
2D structure for PGDB_C002237
GI50-<100nM-GSPT1-HL-60WO2023237116A1PGDB_A013305PGDB_C002237PGDB_AS001555View
2D structure for PGDB_C002218
GI50-=11.38nM-GSPT1-SU-DHL-2WO2023237116A1PGDB_A013438PGDB_C002218PGDB_AS000205View
2D structure for PGDB_C002312
GI50-=100-1000nM-GSPT1-HL-60WO2023237116A1PGDB_A014058PGDB_C002312PGDB_AS001555View
2D structure for PGDB_C002294
GI50-=1000-5000nM-GSPT1-HL-60WO2023237116A1PGDB_A014228PGDB_C002294PGDB_AS001555View
2D structure for PGDB_C002208
GI50-=19.61nM-GSPT1-ToledoWO2023237116A1PGDB_A014474PGDB_C002208PGDB_AS002036View
2D structure for PGDB_C002229
GI50-=0.96nM-GSPT1-ToledoWO2023237116A1PGDB_A014475PGDB_C002229PGDB_AS002036View
2D structure for PGDB_C002220
DC50-<100nM-GSPT1-HEK293WO2023237116A1PGDB_A014996PGDB_C002220PGDB_AS002200View