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Compound
PGDB_C002829
8 activity records1 related patents
2D structure
COc1cc(C(=O)Nc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)ccc1Oc1ccccc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 69.9 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A009809 | PGDB_C002829 | PGDB_AS000685 | View |
| % Degradation | - | = | 17.2 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A019660 | PGDB_C002829 | PGDB_AS000768 | View |
| % Degradation | - | = | 21.3 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A025129 | PGDB_C002829 | PGDB_AS001974 | View |
| % Degradation | - | = | 64.1 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A039647 | PGDB_C002829 | PGDB_AS000209 | View |
| % Degradation | - | = | 81.8 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A049789 | PGDB_C002829 | PGDB_AS001414 | View |
| % Degradation | - | = | 12.1 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A054620 | PGDB_C002829 | PGDB_AS002431 | View |
| % Degradation | - | = | 8.7 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A055433 | PGDB_C002829 | PGDB_AS000707 | View |
| % Degradation | - | = | 92.8 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A072668 | PGDB_C002829 | PGDB_AS000892 | View |