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Compound
PGDB_C002831
8 activity records1 related patents
2D structure
Cc1ccc2c(c1)OCC(C(=O)Nc1ccc3c(c1)CN(C1CCC(=O)NC1=O)C3=O)=C2Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 24 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A007660 | PGDB_C002831 | PGDB_AS000768 | View |
| % Degradation | - | = | 66.9 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A028709 | PGDB_C002831 | PGDB_AS000685 | View |
| % Degradation | - | = | 63.5 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A031383 | PGDB_C002831 | PGDB_AS000209 | View |
| % Degradation | - | = | 28 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A047152 | PGDB_C002831 | PGDB_AS001974 | View |
| % Degradation | - | = | 91.5 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A056781 | PGDB_C002831 | PGDB_AS000892 | View |
| % Degradation | - | = | 72.6 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A065176 | PGDB_C002831 | PGDB_AS001414 | View |
| % Degradation | - | = | 14.3 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A068963 | PGDB_C002831 | PGDB_AS002431 | View |
| % Degradation | - | = | 8.6 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A072168 | PGDB_C002831 | PGDB_AS000707 | View |