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Compound
PGDB_C002835
8 activity records1 related patents
2D structure
COc1ccc2c(c1)OCC(C(=O)Nc1ccc3c(c1)CN(C1CCC(=O)NC1=O)C3=O)=C2Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 32.5 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A019541 | PGDB_C002835 | PGDB_AS000768 | View |
| % Degradation | - | = | 4.3 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A024544 | PGDB_C002835 | PGDB_AS000707 | View |
| % Degradation | - | = | 64.8 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A024568 | PGDB_C002835 | PGDB_AS000685 | View |
| % Degradation | - | = | 59.5 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A025646 | PGDB_C002835 | PGDB_AS000209 | View |
| % Degradation | - | = | 57.1 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A046558 | PGDB_C002835 | PGDB_AS001414 | View |
| % Degradation | - | = | 9 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A050659 | PGDB_C002835 | PGDB_AS002431 | View |
| % Degradation | - | = | 37.5 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A056504 | PGDB_C002835 | PGDB_AS001974 | View |
| % Degradation | - | = | 96 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A067735 | PGDB_C002835 | PGDB_AS000892 | View |