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SIMM · NJU
Assay
PGDB_AS000677
System: cell_based
Target: CDK2
Cell line: HEK293
Assay context summary
Assay context
50 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
CDK2
E3
Not specified
Cell line
HEK293
Technology
luminescence
Activity compounds and values
Activity records
50 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
62
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A009307
PGDB_C007993
PGDB_AS000677
View
Dmax
-
=
79
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A009633
PGDB_C007981
PGDB_AS000677
View
Dmax
-
=
70
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A011631
PGDB_C007996
PGDB_AS000677
View
Dmax
-
=
67
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A016103
PGDB_C007973
PGDB_AS000677
View
Dmax
-
=
50
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A018486
PGDB_C007976
PGDB_AS000677
View
Dmax
-
=
58
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A018813
PGDB_C007986
PGDB_AS000677
View
Dmax
-
=
67
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A020316
PGDB_C007979
PGDB_AS000677
View
Dmax
-
=
65
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A020696
PGDB_C008004
PGDB_AS000677
View
Dmax
-
=
76
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A021741
PGDB_C008016
PGDB_AS000677
View
Dmax
-
=
75
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A021781
PGDB_C008011
PGDB_AS000677
View
Dmax
-
=
66
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A022397
PGDB_C008007
PGDB_AS000677
View
Dmax
-
=
69
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A023089
PGDB_C008015
PGDB_AS000677
View
Dmax
-
=
74
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A023294
PGDB_C007994
PGDB_AS000677
View
Dmax
-
=
58
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A023630
PGDB_C007982
PGDB_AS000677
View
Dmax
-
=
50
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A023800
PGDB_C007970
PGDB_AS000677
View
Dmax
-
=
59
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A023864
PGDB_C007995
PGDB_AS000677
View
Dmax
-
=
67
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A024184
PGDB_C007971
PGDB_AS000677
View
Dmax
-
=
69
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A025254
PGDB_C008000
PGDB_AS000677
View
Dmax
-
=
78
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A026511
PGDB_C008009
PGDB_AS000677
View
Dmax
-
=
79
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A029832
PGDB_C007997
PGDB_AS000677
View