Assay

PGDB_AS001853

System: cell_basedTarget: GSPT1Cell line: HEK293
Assay context summary

Assay context

9 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetGSPT1
E3Not specified
Cell lineHEK293
Detection targetprotein_degradation
Activity compounds and values

Activity records

9 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C001479
DC50-=8.41nM-—GSPT1-HEK293CN118852145APGDB_A032474PGDB_C001479PGDB_AS001853View
2D structure for PGDB_C001471
DC50-=3.24nM-—GSPT1-HEK293CN118852145APGDB_A043485PGDB_C001471PGDB_AS001853View
2D structure for PGDB_C001468
DC50-=1.49nM-—GSPT1-HEK293CN118852145APGDB_A045359PGDB_C001468PGDB_AS001853View
2D structure for PGDB_C001465
DC50-=4.09nM-—GSPT1-HEK293CN118852145APGDB_A056822PGDB_C001465PGDB_AS001853View
2D structure for PGDB_C001474
DC50-=5.64nM-—GSPT1-HEK293CN118852145APGDB_A059678PGDB_C001474PGDB_AS001853View
2D structure for PGDB_C001466
DC50-=4.84nM-—GSPT1-HEK293CN118852145APGDB_A060495PGDB_C001466PGDB_AS001853View
2D structure for PGDB_C001470
DC50-=1.67nM-—GSPT1-HEK293CN118852145APGDB_A069918PGDB_C001470PGDB_AS001853View
2D structure for PGDB_C001475
DC50-=5nM-—GSPT1-HEK293CN118852145APGDB_A073744PGDB_C001475PGDB_AS001853View
2D structure for PGDB_C001478
DC50-=3.71nM-—GSPT1-HEK293CN118852145APGDB_A076182PGDB_C001478PGDB_AS001853View
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