Assay context summary

Assay context

55 activity records
Activity compounds and values

Activity records

55 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C001313
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A008470PGDB_C001313PGDB_AS002288View
2D structure for PGDB_C001343
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A008905PGDB_C001343PGDB_AS002288View
2D structure for PGDB_C001351
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A009661PGDB_C001351PGDB_AS002288View
2D structure for PGDB_C001338
% Degradation-=30-50%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A010299PGDB_C001338PGDB_AS002288View
2D structure for PGDB_C001349
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A011451PGDB_C001349PGDB_AS002288View
2D structure for PGDB_C001322
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A014409PGDB_C001322PGDB_AS002288View
2D structure for PGDB_C001341
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A014772PGDB_C001341PGDB_AS002288View
2D structure for PGDB_C001339
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A015977PGDB_C001339PGDB_AS002288View
2D structure for PGDB_C001348
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A016250PGDB_C001348PGDB_AS002288View
2D structure for PGDB_C001318
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A016876PGDB_C001318PGDB_AS002288View
2D structure for PGDB_C001356
% Degradation-<=30%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A017183PGDB_C001356PGDB_AS002288View
2D structure for PGDB_C001355
% Degradation-=50-70%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A019398PGDB_C001355PGDB_AS002288View
2D structure for PGDB_C001312
% Degradation-=50-70%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A020051PGDB_C001312PGDB_AS002288View
2D structure for PGDB_C001329
% Degradation-=30-50%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A021689PGDB_C001329PGDB_AS002288View
2D structure for PGDB_C001324
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A025304PGDB_C001324PGDB_AS002288View
2D structure for PGDB_C001359
% Degradation-<=30%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A025411PGDB_C001359PGDB_AS002288View
2D structure for PGDB_C001301
% Degradation-=30-50%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A027617PGDB_C001301PGDB_AS002288View
2D structure for PGDB_C001332
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A028199PGDB_C001332PGDB_AS002288View
2D structure for PGDB_C001321
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A031387PGDB_C001321PGDB_AS002288View
2D structure for PGDB_C001344
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatKR20250075510APGDB_A031484PGDB_C001344PGDB_AS002288View