Summary
AssigneeFudan University
Filing years2022
Patents1
Compounds66
Activity records185
Patent families1
Targets1
Assay familiesdegradation, viability
Activity metricsIC50, degradation
Overview

Target distribution and active-compound trend

Target distribution

185 activity records

1 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

033662024
Activity compounds and values

Activity records

185 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C005341
% Degradation-=38.1%--GSPT1-JeKo-1WO2023078410A1PGDB_A008346PGDB_C005341PGDB_AS002119View
2D structure for PGDB_C005320
% Degradation-=56%--GSPT1-JeKo-1WO2023078410A1PGDB_A008510PGDB_C005320PGDB_AS000305View
2D structure for PGDB_C005331
IC50-=11.6nM-GSPT1-HL-60WO2023078410A1PGDB_A008888PGDB_C005331PGDB_AS002047View
2D structure for PGDB_C005356
% Degradation-=11.6%--GSPT1-JeKo-1WO2023078410A1PGDB_A009031PGDB_C005356PGDB_AS002119View
2D structure for PGDB_C005331
% Degradation-=95%--GSPT1-JeKo-1WO2023078410A1PGDB_A009617PGDB_C005331PGDB_AS000305View
2D structure for PGDB_C005311
% Degradation-=97%--GSPT1-JeKo-1WO2023078410A1PGDB_A009651PGDB_C005311PGDB_AS000305View
2D structure for PGDB_C005315
% Degradation-=33%--GSPT1-JeKo-1WO2023078410A1PGDB_A009788PGDB_C005315PGDB_AS002119View
2D structure for PGDB_C005327
IC50-=14.3nM-GSPT1-HL-60WO2023078410A1PGDB_A010274PGDB_C005327PGDB_AS002047View
2D structure for PGDB_C005329
% Degradation-=95.6%--GSPT1-JeKo-1WO2023078410A1PGDB_A012097PGDB_C005329PGDB_AS000305View
2D structure for PGDB_C005308
IC50-=6.2nM-GSPT1-HNT-34WO2023078410A1PGDB_A014569PGDB_C005308PGDB_AS000001View
2D structure for PGDB_C005300
IC50-=26.9nM-GSPT1-HNT-34WO2023078410A1PGDB_A014587PGDB_C005300PGDB_AS000001View
2D structure for PGDB_C005328
% Degradation-=100%--GSPT1-JeKo-1WO2023078410A1PGDB_A014777PGDB_C005328PGDB_AS002119View
2D structure for PGDB_C005322
% Degradation-=96%--GSPT1-JeKo-1WO2023078410A1PGDB_A014797PGDB_C005322PGDB_AS002119View
2D structure for PGDB_C005323
% Degradation-=93%--GSPT1-JeKo-1WO2023078410A1PGDB_A015297PGDB_C005323PGDB_AS002119View
2D structure for PGDB_C005302
% Degradation-=97%--GSPT1-JeKo-1WO2023078410A1PGDB_A015727PGDB_C005302PGDB_AS000305View
2D structure for PGDB_C005355
% Degradation-=77.7%--GSPT1-JeKo-1WO2023078410A1PGDB_A015736PGDB_C005355PGDB_AS002119View
2D structure for PGDB_C005351
% Degradation-=96.2%--GSPT1-JeKo-1WO2023078410A1PGDB_A016297PGDB_C005351PGDB_AS002119View
2D structure for PGDB_C005340
% Degradation-=80%--GSPT1-JeKo-1WO2023078410A1PGDB_A016595PGDB_C005340PGDB_AS000305View
2D structure for PGDB_C005313
% Degradation-=77%--GSPT1-JeKo-1WO2023078410A1PGDB_A016833PGDB_C005313PGDB_AS000305View
2D structure for PGDB_C005345
% Degradation-=51%--GSPT1-JeKo-1WO2023078410A1PGDB_A016861PGDB_C005345PGDB_AS002119View