Assignee profile

Ileadbms

Coverage of patents, compounds and activity records linked to this assignee.

1 patents109 compounds325 activity records
Summary
AssigneeIleadbms
Filing years2024
Patents1
Compounds109
Activity records325
Patent families1
Targets3
Assay familiesdegradation
Activity metricsIC50
Overview

Target distribution and active-compound trend

Target distribution

545 activity records

4 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

0551092025
Activity compounds and values

Activity records

545 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C010919
IC50-<=0.1uM-—CDK13--WO2025110815A1PGDB_A007078PGDB_C010919PGDB_AS001146View
2D structure for PGDB_C010990
IC50-<=0.3uM-—POLR2A--WO2025110815A1PGDB_A007136PGDB_C010990PGDB_AS000589View
2D structure for PGDB_C010931
IC50-=0.05-0.5uM-—--MDA-MB-231WO2025110815A1PGDB_A007260PGDB_C010931PGDB_AS000344View
2D structure for PGDB_C010927
IC50->0.5uM-—--MDA-MB-231WO2025110815A1PGDB_A007382PGDB_C010927PGDB_AS000344View
2D structure for PGDB_C010967
IC50-<=0.1uM-—CDK13--WO2025110815A1PGDB_A007659PGDB_C010967PGDB_AS001146View
2D structure for PGDB_C010941
IC50-<=0.1uM-—CDK12--WO2025110815A1PGDB_A007735PGDB_C010941PGDB_AS002095View
2D structure for PGDB_C010952
Selectivity index-=100-500fold-—---WO2025110815A1PGDB_A007998PGDB_C010952PGDB_AS002417View
2D structure for PGDB_C010923
IC50-=0.1-0.5uM-—CDK13--WO2025110815A1PGDB_A008213PGDB_C010923PGDB_AS001146View
2D structure for PGDB_C010982
IC50-<=0.05uM-—--MDA-MB-231WO2025110815A1PGDB_A008242PGDB_C010982PGDB_AS000344View
2D structure for PGDB_C010965
IC50-=0.3-3uM-—POLR2A--WO2025110815A1PGDB_A008267PGDB_C010965PGDB_AS000589View
2D structure for PGDB_C011002
IC50-<=0.3uM-—POLR2A--WO2025110815A1PGDB_A008324PGDB_C011002PGDB_AS000589View
2D structure for PGDB_C010960
Selectivity index->500fold-—---WO2025110815A1PGDB_A008572PGDB_C010960PGDB_AS002417View
2D structure for PGDB_C010920
Selectivity index->500fold-—---WO2025110815A1PGDB_A008916PGDB_C010920PGDB_AS002417View
2D structure for PGDB_C010943
IC50-<=0.2uM-—--MKN1WO2025110815A1PGDB_A008972PGDB_C010943PGDB_AS000785View
2D structure for PGDB_C010924
IC50->0.5uM-—--MDA-MB-231WO2025110815A1PGDB_A009022PGDB_C010924PGDB_AS000344View
2D structure for PGDB_C010921
IC50-<=0.3uM-—POLR2A--WO2025110815A1PGDB_A009103PGDB_C010921PGDB_AS000589View
2D structure for PGDB_C011000
IC50-<=0.3uM-—POLR2A--WO2025110815A1PGDB_A009351PGDB_C011000PGDB_AS000589View
2D structure for PGDB_C010902
IC50-<=0.2uM-—--SW480WO2025110815A1PGDB_A009579PGDB_C010902PGDB_AS002136View
2D structure for PGDB_C010977
IC50-<=0.1uM-—CDK13--WO2025110815A1PGDB_A009848PGDB_C010977PGDB_AS001146View
2D structure for PGDB_C010929
IC50->3uM-—POLR2A--WO2025110815A1PGDB_A009975PGDB_C010929PGDB_AS000589View
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