Summary
AssigneeShanghai Qilu Pharmaceutical Research And Development Centre
Filing years2025
Patents2
Compounds322
Activity records764
Patent families2
Targets2
Assay familiesdegradation, viability
Activity metricsDC50, Dmax, IC50
Overview

Target distribution and active-compound trend

Target distribution

762 activity records

2 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

013827520252026
Activity compounds and values

Activity records

762 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C005465
IC50-=20.27nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A007288PGDB_C005465PGDB_AS001340View
2D structure for PGDB_C005474
DC50-=6.12nM-GSPT1-HEK293WO2025252247A1PGDB_A009168PGDB_C005474PGDB_AS000196View
2D structure for PGDB_C005479
IC50-=14.99nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A009609PGDB_C005479PGDB_AS000582View
2D structure for PGDB_C005468
IC50-=22.92nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A010357PGDB_C005468PGDB_AS001340View
2D structure for PGDB_C005496
IC50-=14.06nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A010402PGDB_C005496PGDB_AS000582View
2D structure for PGDB_C005502
IC50-=40.39nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A010559PGDB_C005502PGDB_AS000582View
2D structure for PGDB_C003382
IC50-=62.69nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A010893PGDB_C003382PGDB_AS000582View
2D structure for PGDB_C005462
IC50-=78.93nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A011256PGDB_C005462PGDB_AS001340View
2D structure for PGDB_C005472
IC50-=25.94nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A012477PGDB_C005472PGDB_AS001340View
2D structure for PGDB_C005486
IC50-=11.36nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A016912PGDB_C005486PGDB_AS000582View
2D structure for PGDB_C005478
IC50-=10.08nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A017687PGDB_C005478PGDB_AS000582View
2D structure for PGDB_C005501
IC50-=90.69nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A017968PGDB_C005501PGDB_AS000582View
2D structure for PGDB_C005481
IC50-=58.39nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A018407PGDB_C005481PGDB_AS000582View
2D structure for PGDB_C005490
IC50-=23.11nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A021436PGDB_C005490PGDB_AS000582View
2D structure for PGDB_C005469
IC50-=98.66nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A022285PGDB_C005469PGDB_AS001340View
2D structure for PGDB_C005497
IC50-=13.91nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A024792PGDB_C005497PGDB_AS000582View
2D structure for PGDB_C003382
IC50-=121.46nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A024823PGDB_C003382PGDB_AS001340View
2D structure for PGDB_C005473
DC50-=2.5nM-GSPT1-HEK293WO2025252247A1PGDB_A025347PGDB_C005473PGDB_AS000196View
2D structure for PGDB_C005468
DC50-=4.9nM-GSPT1-HEK293WO2025252247A1PGDB_A031373PGDB_C005468PGDB_AS000196View
2D structure for PGDB_C005506
IC50-=18.43nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A032172PGDB_C005506PGDB_AS000582View