Assay context summary

Assay context

216 activity records
Activity compounds and values

Activity records

216 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C024203
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A007023PGDB_C024203PGDB_AS000351View
2D structure for PGDB_C024407
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A007292PGDB_C024407PGDB_AS000351View
2D structure for PGDB_C024427
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A008275PGDB_C024427PGDB_AS000351View
2D structure for PGDB_C024450
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A008672PGDB_C024450PGDB_AS000351View
2D structure for PGDB_C024447
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A008696PGDB_C024447PGDB_AS000351View
2D structure for PGDB_C024345
% Degradation-=20-100%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A008851PGDB_C024345PGDB_AS000351View
2D structure for PGDB_C024330
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A008977PGDB_C024330PGDB_AS000351View
2D structure for PGDB_C024433
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A009393PGDB_C024433PGDB_AS000351View
2D structure for PGDB_C024366
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A009844PGDB_C024366PGDB_AS000351View
2D structure for PGDB_C024380
% Degradation-=20-100%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A010113PGDB_C024380PGDB_AS000351View
2D structure for PGDB_C024227
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A010153PGDB_C024227PGDB_AS000351View
2D structure for PGDB_C024416
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A010196PGDB_C024416PGDB_AS000351View
2D structure for PGDB_C024437
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A010277PGDB_C024437PGDB_AS000351View
2D structure for PGDB_C024443
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A010329PGDB_C024443PGDB_AS000351View
2D structure for PGDB_C024247
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A010453PGDB_C024247PGDB_AS000351View
2D structure for PGDB_C024395
% Degradation-=20-100%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A010840PGDB_C024395PGDB_AS000351View
2D structure for PGDB_C024319
% Degradation-=20-100%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A011097PGDB_C024319PGDB_AS000351View
2D structure for PGDB_C024414
% Degradation-=20-100%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A012690PGDB_C024414PGDB_AS000351View
2D structure for PGDB_C024436
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A013250PGDB_C024436PGDB_AS000351View
2D structure for PGDB_C024281
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--WO2025162225A1PGDB_A013471PGDB_C024281PGDB_AS000351View