Assay

PGDB_AS002309

System: cell_basedTarget: CDK2Cell line: HEK293
Assay context summary

Assay context

30 activity records
Assay family% Degradation
Systemcell_based
ReadoutIC50
TargetCDK2
E3Not specified
Cell lineHEK293
Technologyluminescence
Activity compounds and values

Activity records

30 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C007943
IC50-=0.079uM-—CDK2-HEK293WO2025043225PGDB_A009413PGDB_C007943PGDB_AS002309View
2D structure for PGDB_C007944
IC50-=0.18uM-—CDK2-HEK293WO2025043225PGDB_A010158PGDB_C007944PGDB_AS002309View
2D structure for PGDB_C007934
IC50-=0.81uM-—CDK2-HEK293WO2025043225PGDB_A011267PGDB_C007934PGDB_AS002309View
2D structure for PGDB_C007939
IC50-=0.18uM-—CDK2-HEK293WO2025043225PGDB_A011923PGDB_C007939PGDB_AS002309View
2D structure for PGDB_C007946
IC50-=0.42uM-—CDK2-HEK293WO2025043225PGDB_A018343PGDB_C007946PGDB_AS002309View
2D structure for PGDB_C007945
IC50-=0.17uM-—CDK2-HEK293WO2025043225PGDB_A020055PGDB_C007945PGDB_AS002309View
2D structure for PGDB_C007951
IC50-=0.49uM-—CDK2-HEK293WO2025043225PGDB_A020729PGDB_C007951PGDB_AS002309View
2D structure for PGDB_C007932
IC50-=0.76uM-—CDK2-HEK293WO2025043225PGDB_A027206PGDB_C007932PGDB_AS002309View
2D structure for PGDB_C007948
IC50-=0.066uM-—CDK2-HEK293WO2025043225PGDB_A030890PGDB_C007948PGDB_AS002309View
2D structure for PGDB_C007933
IC50-=0.11uM-—CDK2-HEK293WO2025043225PGDB_A033143PGDB_C007933PGDB_AS002309View
2D structure for PGDB_C007941
IC50-=0.16uM-—CDK2-HEK293WO2025043225PGDB_A033591PGDB_C007941PGDB_AS002309View
2D structure for PGDB_C007935
IC50-=0.15uM-—CDK2-HEK293WO2025043225PGDB_A034508PGDB_C007935PGDB_AS002309View
2D structure for PGDB_C007957
IC50-=0.16uM-—CDK2-HEK293WO2025043225PGDB_A040936PGDB_C007957PGDB_AS002309View
2D structure for PGDB_C007942
IC50-=0.12uM-—CDK2-HEK293WO2025043225PGDB_A045674PGDB_C007942PGDB_AS002309View
2D structure for PGDB_C007952
IC50-=0.58uM-—CDK2-HEK293WO2025043225PGDB_A050038PGDB_C007952PGDB_AS002309View
2D structure for PGDB_C007940
IC50-=0.26uM-—CDK2-HEK293WO2025043225PGDB_A050255PGDB_C007940PGDB_AS002309View
2D structure for PGDB_C007953
IC50-=0.44uM-—CDK2-HEK293WO2025043225PGDB_A050398PGDB_C007953PGDB_AS002309View
2D structure for PGDB_C007955
IC50-=0.12uM-—CDK2-HEK293WO2025043225PGDB_A055133PGDB_C007955PGDB_AS002309View
2D structure for PGDB_C007956
IC50-=0.2uM-—CDK2-HEK293WO2025043225PGDB_A056239PGDB_C007956PGDB_AS002309View
2D structure for PGDB_C007937
IC50-=1.1uM-—CDK2-HEK293WO2025043225PGDB_A060090PGDB_C007937PGDB_AS002309View
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