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SIMM · NJU
Assay
PGDB_AS001468
System: cell_based
Target: CDK2
Cell line: HEK293
Assay context summary
Assay context
30 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
CDK2
E3
Not specified
Cell line
HEK293
Technology
luminescence
Activity compounds and values
Activity records
30 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
49
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A013106
PGDB_C007948
PGDB_AS001468
View
Dmax
-
=
28
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A015684
PGDB_C007933
PGDB_AS001468
View
Dmax
-
=
26
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A016686
PGDB_C007932
PGDB_AS001468
View
Dmax
-
=
17
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A017087
PGDB_C007955
PGDB_AS001468
View
Dmax
-
=
32
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A018753
PGDB_C007942
PGDB_AS001468
View
Dmax
-
=
27
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A020423
PGDB_C007945
PGDB_AS001468
View
Dmax
-
=
42
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A021560
PGDB_C007936
PGDB_AS001468
View
Dmax
-
=
26
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A024771
PGDB_C007961
PGDB_AS001468
View
Dmax
-
=
29
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A025075
PGDB_C007937
PGDB_AS001468
View
Dmax
-
=
24
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A026678
PGDB_C007941
PGDB_AS001468
View
Dmax
-
=
22
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A028745
PGDB_C007958
PGDB_AS001468
View
Dmax
-
=
45
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A029566
PGDB_C007935
PGDB_AS001468
View
Dmax
-
=
26
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A035515
PGDB_C007957
PGDB_AS001468
View
Dmax
-
=
33
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A037128
PGDB_C007947
PGDB_AS001468
View
Dmax
-
=
27
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A037581
PGDB_C007956
PGDB_AS001468
View
Dmax
-
=
47
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A038625
PGDB_C007934
PGDB_AS001468
View
Dmax
-
=
12
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A039405
PGDB_C007954
PGDB_AS001468
View
Dmax
-
=
35
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A041025
PGDB_C007950
PGDB_AS001468
View
Dmax
-
=
22
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A048865
PGDB_C007940
PGDB_AS001468
View
Dmax
-
=
17
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A051428
PGDB_C007944
PGDB_AS001468
View