Summary
AssigneeProtier Biotech
Filing years2024
Patents1
Compounds60
Activity records269
Patent families1
Targets2
Assay familiesbinding, degradation, viability
Activity metricsGI50, degradation, relative_binding
Overview

Target distribution and active-compound trend

Target distribution

269 activity records

2 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

030602025
Activity compounds and values

Activity records

269 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C001322
% Degradation-=90-100%--GSPT1-JurkatWO2025110699A1PGDB_A007052PGDB_C001322PGDB_AS001994View
2D structure for PGDB_C001336
% Degradation-=70-90%--GSPT1-JurkatWO2025110699A1PGDB_A007081PGDB_C001336PGDB_AS001067View
2D structure for PGDB_C001345
% Degradation-=70-90%--GSPT1-JurkatWO2025110699A1PGDB_A007788PGDB_C001345PGDB_AS001994View
2D structure for PGDB_C001302
% Degradation-=90-100%--GSPT1-JurkatWO2025110699A1PGDB_A008236PGDB_C001302PGDB_AS001067View
2D structure for PGDB_C001312
GI50-=0.1-1uM-GSPT1-JurkatWO2025110699A1PGDB_A008601PGDB_C001312PGDB_AS001887View
2D structure for PGDB_C001329
% Degradation-=30-50%--GSPT1-JurkatWO2025110699A1PGDB_A008778PGDB_C001329PGDB_AS001067View
2D structure for PGDB_C001317
% Degradation-=50-70%--GSPT1-JurkatWO2025110699A1PGDB_A009275PGDB_C001317PGDB_AS001008View
2D structure for PGDB_C001327
GI50-<=0.1uM-GSPT1-MM.1SWO2025110699A1PGDB_A009373PGDB_C001327PGDB_AS002497View
2D structure for PGDB_C001330
% Degradation-=90-100%--GSPT1-JurkatWO2025110699A1PGDB_A009427PGDB_C001330PGDB_AS001994View
2D structure for PGDB_C001348
GI50-=0.1-1uM-GSPT1-JurkatWO2025110699A1PGDB_A010010PGDB_C001348PGDB_AS001887View
2D structure for PGDB_C001336
% Degradation-=70-90%--GSPT1-JurkatWO2025110699A1PGDB_A010367PGDB_C001336PGDB_AS001008View
2D structure for PGDB_C001326
GI50-<=0.1uM-GSPT1-JurkatWO2025110699A1PGDB_A010463PGDB_C001326PGDB_AS001887View
2D structure for PGDB_C001340
% Degradation-=50-70%--GSPT1-JurkatWO2025110699A1PGDB_A010634PGDB_C001340PGDB_AS001067View
2D structure for PGDB_C001303
Relative binding-<1%--CRBNCRBNHEK293WO2025110699A1PGDB_A011004PGDB_C001303PGDB_AS001966View
2D structure for PGDB_C001314
Relative binding-<0.1%--CRBNCRBNHEK293WO2025110699A1PGDB_A011063PGDB_C001314PGDB_AS001966View
2D structure for PGDB_C001325
GI50-<=0.1uM-GSPT1-MM.1SWO2025110699A1PGDB_A011311PGDB_C001325PGDB_AS002497View
2D structure for PGDB_C001349
% Degradation-=90-100%--GSPT1-JurkatWO2025110699A1PGDB_A011384PGDB_C001349PGDB_AS001008View
2D structure for PGDB_C001344
% Degradation-=70-90%--GSPT1-JurkatWO2025110699A1PGDB_A011460PGDB_C001344PGDB_AS001008View
2D structure for PGDB_C001321
% Degradation-=90-100%--GSPT1-JurkatWO2025110699A1PGDB_A011515PGDB_C001321PGDB_AS001008View
2D structure for PGDB_C001348
% Degradation-=90-100%--GSPT1-JurkatWO2025110699A1PGDB_A012657PGDB_C001348PGDB_AS001008View