Summary
AssigneeHarvard University
Filing years2023
Patents1
Compounds44
Activity records398
Patent families1
Targets4
Assay familiesdegradation
Activity metricsDC50, Dmax, degradation
Overview

Target distribution and active-compound trend

Target distribution

398 activity records

4 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

022442024
Activity compounds and values

Activity records

398 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C002810
% Degradation-=67.4%--CSNK1A1--WO2024059107A1PGDB_A007173PGDB_C002810PGDB_AS000685View
2D structure for PGDB_C002807
% Degradation-=4.4%--IKZF1--WO2024059107A1PGDB_A007445PGDB_C002807PGDB_AS000707View
2D structure for PGDB_C002831
% Degradation-=24%--IKZF1--WO2024059107A1PGDB_A007660PGDB_C002831PGDB_AS000768View
2D structure for PGDB_C002837
% Degradation-=6.1%--GSPT1--WO2024059107A1PGDB_A008001PGDB_C002837PGDB_AS002431View
2D structure for PGDB_C002828
% Degradation-=7%--IKZF1--WO2024059107A1PGDB_A008146PGDB_C002828PGDB_AS000768View
2D structure for PGDB_C002813
% Degradation-=55.4%--CSNK1A1--WO2024059107A1PGDB_A008181PGDB_C002813PGDB_AS000685View
2D structure for PGDB_C002813
% Degradation-=9.3%--IKZF1--WO2024059107A1PGDB_A008209PGDB_C002813PGDB_AS000707View
2D structure for PGDB_C002847
Dmax-=40.3%--CSNK1A1--WO2024059107A1PGDB_A008277PGDB_C002847PGDB_AS002567View
2D structure for PGDB_C002826
% Degradation-=12.5%--GSPT1--WO2024059107A1PGDB_A008406PGDB_C002826PGDB_AS002431View
2D structure for PGDB_C002845
Dmax-=92.8%--IKZF2-NCI-H1155WO2024059107A1PGDB_A008488PGDB_C002845PGDB_AS000259View
2D structure for PGDB_C002817
% Degradation-=70.8%--IKZF2--WO2024059107A1PGDB_A008495PGDB_C002817PGDB_AS001414View
2D structure for PGDB_C002849
DC50-=72nM-IKZF1-NCI-H1155WO2024059107A1PGDB_A008514PGDB_C002849PGDB_AS001115View
2D structure for PGDB_C002834
% Degradation-=75%--IKZF2--WO2024059107A1PGDB_A008953PGDB_C002834PGDB_AS001414View
2D structure for PGDB_C002819
% Degradation-=50.2%--CSNK1A1--WO2024059107A1PGDB_A009085PGDB_C002819PGDB_AS000209View
2D structure for PGDB_C002834
% Degradation-=9.2%--GSPT1--WO2024059107A1PGDB_A009147PGDB_C002834PGDB_AS002431View
2D structure for PGDB_C002843
% Degradation-=76.2%--CSNK1A1--WO2024059107A1PGDB_A009175PGDB_C002843PGDB_AS000209View
2D structure for PGDB_C002838
% Degradation-=91.8%--IKZF2--WO2024059107A1PGDB_A009399PGDB_C002838PGDB_AS000892View
2D structure for PGDB_C002828
% Degradation-=48.1%--CSNK1A1--WO2024059107A1PGDB_A009504PGDB_C002828PGDB_AS000209View
2D structure for PGDB_C002829
% Degradation-=69.9%--CSNK1A1--WO2024059107A1PGDB_A009809PGDB_C002829PGDB_AS000685View
2D structure for PGDB_C002845
% Degradation-=51.3%--CSNK1A1--WO2024059107A1PGDB_A010007PGDB_C002845PGDB_AS000209View