Browse
Targets
| Compounds | Activity records | Details | ||
|---|---|---|---|---|
| CRBN | E3_ligase | assay_marker | 5504 | 10585 | View |
| GSPT1 | assay_context_marker | assay_marker | degradation_target | effector | neo_substrate | primary_target | 5338 | 8048 | View |
| IKZF2 | assay_marker | degradation_target | neo_substrate | primary_target | 3288 | 5896 | View |
| IKZF1 | assay_marker | degradation_target | neo_substrate | primary_target | 3340 | 4601 | View |
| SMARCA2 | degradation_target | primary_target | 1496 | 3232 | View |
| CSNK1A1 | degradation_target | neo_substrate | primary_target | 2064 | 3065 | View |
| SMARCA4 | degradation_target | primary_target | 1400 | 2955 | View |
| WEE1 | degradation_target | neo_substrate | primary_target | 2074 | 2842 | View |
| VAV1 | degradation_target | primary_target | 1241 | 2475 | View |
| DDB1 | E3_complex_component | E3_ligase | binding_target | effector | primary_target | 1829 | 2443 | View |
| AR | degradation_target | primary_target | 481 | 2219 | View |
| IKZF3 | assay_marker | degradation_target | neo_substrate | primary_target | 1616 | 2170 | View |
| NEK7 | degradation_target | neo_substrate | primary_target | 478 | 1960 | View |
| KRAS | binding_partner | degradation_target | primary_target | 544 | 1802 | View |
| CDK2 | assay_marker | degradation_target | primary_target | 548 | 1000 | View |
| DCAF15 | E3_ligase | effector | primary_target | 521 | 827 | View |
| SKP1 | E3_complex_component | 349 | 685 | View |
| FBXW11 | E3_ligase | 349 | 685 | View |
| BTRC | E3_ligase | 349 | 685 | View |
| ALK | degradation_target | primary_target | 209 | 650 | View |
| CCNK | assay_complex_component | degradation_target | neo_substrate | primary_target | 438 | 604 | View |
| BRAF | degradation_target | effector | primary_target | 251 | 553 | View |
| RBM39 | degradation_target | neo_substrate | primary_target | 521 | 535 | View |
| CDK12 | primary_target | 180 | 515 | View |
| MYC | degradation_target | neo_substrate | primary_target | 310 | 430 | View |