Assay context summary

Assay context

20 activity records
Activity compounds and values

Activity records

20 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C024266
% Inhibition-=50-60%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A018174PGDB_C024266PGDB_AS002558View
2D structure for PGDB_C024255
% Inhibition-=40-50%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A018551PGDB_C024255PGDB_AS002558View
2D structure for PGDB_C024211
% Inhibition-=70-80%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A020805PGDB_C024211PGDB_AS002558View
2D structure for PGDB_C024265
% Inhibition-=40-50%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A027335PGDB_C024265PGDB_AS002558View
2D structure for PGDB_C024215
% Inhibition-=50-60%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A031124PGDB_C024215PGDB_AS002558View
2D structure for PGDB_C024193
% Inhibition-=50-60%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A034813PGDB_C024193PGDB_AS002558View
2D structure for PGDB_C024195
% Inhibition-=80-100%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A035238PGDB_C024195PGDB_AS002558View
2D structure for PGDB_C024262
% Inhibition-=60-70%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A041027PGDB_C024262PGDB_AS002558View
2D structure for PGDB_C024194
% Inhibition-=70-80%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A042462PGDB_C024194PGDB_AS002558View
2D structure for PGDB_C024261
% Inhibition-=40-50%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A050453PGDB_C024261PGDB_AS002558View
2D structure for PGDB_C024264
% Inhibition-=60-70%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A052614PGDB_C024264PGDB_AS002558View
2D structure for PGDB_C024260
% Inhibition-=40-50%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A054488PGDB_C024260PGDB_AS002558View
2D structure for PGDB_C024257
% Inhibition-=50-60%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A055589PGDB_C024257PGDB_AS002558View
2D structure for PGDB_C024244
% Inhibition-=40-50%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A057858PGDB_C024244PGDB_AS002558View
2D structure for PGDB_C024192
% Inhibition-=40-50%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A058626PGDB_C024192PGDB_AS002558View
2D structure for PGDB_C024263
% Inhibition-=60-70%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A065393PGDB_C024263PGDB_AS002558View
2D structure for PGDB_C024254
% Inhibition-=60-70%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A067171PGDB_C024254PGDB_AS002558View
2D structure for PGDB_C024258
% Inhibition-=70-80%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A071838PGDB_C024258PGDB_AS002558View
2D structure for PGDB_C024256
% Inhibition-=60-70%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A074242PGDB_C024256PGDB_AS002558View
2D structure for PGDB_C024259
% Inhibition-=50-60%500 nM96 hIKZF3-TMD8WO2025162225A1PGDB_A076193PGDB_C024259PGDB_AS002558View