Summary
AssigneeScripps Research Institute
Filing years2019
Patents1
Compounds62
Activity records528
Patent families1
Targets2
Assay familiesbiochemical
Activity metricsDmax, EC50
Overview

Target distribution and active-compound trend

Target distribution

528 activity records

2 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

031622019
Activity compounds and values

Activity records

528 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C019895
EC50-=0.0000000089M-CYCEP--WO2019200310A1PGDB_A007025PGDB_C019895PGDB_AS001078View
2D structure for PGDB_C019882
EC50-=0.0000142M-FBXW7--WO2019200310A1PGDB_A007266PGDB_C019882PGDB_AS002126View
2D structure for PGDB_C021159
EC50-=0.0000022M-FBXW7--WO2019200310A1PGDB_A007401PGDB_C021159PGDB_AS002126View
2D structure for PGDB_C019915
EC50-=0.0000127M-FBXW7--WO2019200310A1PGDB_A007442PGDB_C019915PGDB_AS000046View
2D structure for PGDB_C019896
EC50-=0.0000653M-FBXW7--WO2019200310A1PGDB_A007624PGDB_C019896PGDB_AS001009View
2D structure for PGDB_C019897
EC50-=0.0000000032M-FBXW7--WO2019200310A1PGDB_A007727PGDB_C019897PGDB_AS000046View
2D structure for PGDB_C019868
EC50-=0.0000754M-FBXW7--WO2019200310A1PGDB_A008024PGDB_C019868PGDB_AS001009View
2D structure for PGDB_C019883
EC50-=0.0000000001318M-FBXW7--WO2019200310A1PGDB_A008072PGDB_C019883PGDB_AS002126View
2D structure for PGDB_C019880
EC50-=0.0000196M-FBXW7--WO2019200310A1PGDB_A008208PGDB_C019880PGDB_AS000046View
2D structure for PGDB_C019904
Dmax-=8.63%--FBXW7--WO2019200310A1PGDB_A008227PGDB_C019904PGDB_AS001280View
2D structure for PGDB_C019887
EC50-=0.0000000203M-FBXW7--WO2019200310A1PGDB_A008602PGDB_C019887PGDB_AS002126View
2D structure for PGDB_C019889
EC50-=0.0000653M-FBXW7--WO2019200310A1PGDB_A008738PGDB_C019889PGDB_AS001009View
2D structure for PGDB_C019874
EC50-=0.0000715M-FBXW7--WO2019200310A1PGDB_A008763PGDB_C019874PGDB_AS000046View
2D structure for PGDB_C019911
EC50-=0.000002M-CYCEP--WO2019200310A1PGDB_A008783PGDB_C019911PGDB_AS001078View
2D structure for PGDB_C019914
EC50-=0.0000593M-FBXW7--WO2019200310A1PGDB_A009057PGDB_C019914PGDB_AS002246View
2D structure for PGDB_C019894
EC50-=0.0000164M-FBXW7--WO2019200310A1PGDB_A009201PGDB_C019894PGDB_AS002126View
2D structure for PGDB_C019917
EC50-=0.0000000903M-FBXW7--WO2019200310A1PGDB_A009207PGDB_C019917PGDB_AS000046View
2D structure for PGDB_C019900
EC50-=0.0000241M-FBXW7--WO2019200310A1PGDB_A009333PGDB_C019900PGDB_AS002126View
2D structure for PGDB_C019903
EC50-=0.0000238M-FBXW7--WO2019200310A1PGDB_A009365PGDB_C019903PGDB_AS000046View
2D structure for PGDB_C019919
Dmax-=0.18%--FBXW7--WO2019200310A1PGDB_A009592PGDB_C019919PGDB_AS000856View